Subtle Changes in Residue 77 of the γ Subunit of α1β2γ2 GABAA Receptors Drastically Alter the Affinity for Ligands of the Benzodiazepine Binding Site - ScienceDirect
Different Residues in the GABAA Receptor Benzodiazepine Binding Pocket Mediate Benzodiazepine Efficacy and Binding | Molecular Pharmacology
IJMS | Free Full-Text | GABAA Receptor Ligands Often Interact with Binding Sites in the Transmembrane Domain and in the Extracellular Domain—Can the Promiscuity Code Be Cracked?
Diazepam-bound GABAA receptor models identify new benzodiazepine binding- site ligands | Nature Chemical Biology
Flavonoids as GABAA receptor ligands: the whole story? - Abstract - Europe PMC
A Unified Model of the GABAA Receptor Comprising Agonist and Benzodiazepine Binding Sites | PLOS ONE
GABAA receptor - Wikipedia
Biomolecules | Free Full-Text | Benzodiazepine Modulation of GABAA Receptors: A Mechanistic Perspective
Structure of a human synaptic GABAA receptor. - Abstract - Europe PMC
Mechanism of Action of the Benzodiazepines - Neurotorium
Subtype Selective γ-Aminobutyric Acid Type A Receptor (GABAAR) Modulators Acting at the Benzodiazepine Binding Site: An Update | Journal of Medicinal Chemistry
Mechanisms Underlying Tolerance after Long-Term Benzodiazepine Use: A Future for Subtype-Selective G A B A A Receptor Modulators?
Two different benzodiazepine-binding sites in ELIC. ( A ) Cross-section... | Download Scientific Diagram
A Unified Model of the GABAA Receptor Comprising Agonist and Benzodiazepine Binding Sites | PLOS ONE
Structure of the GABAA receptor (side and top views)'" and position of... | Download Scientific Diagram
Frontiers | The Z-Drugs Zolpidem, Zaleplon, and Eszopiclone Have Varying Actions on Human GABAA Receptors Containing γ1, γ2, and γ3 Subunits
IJMS | Free Full-Text | GABAA Receptor Ligands Often Interact with Binding Sites in the Transmembrane Domain and in the Extracellular Domain—Can the Promiscuity Code Be Cracked?
GABAA receptor - Wikipedia
The GABAA receptor and benzodiazepine acceptor site
Sedative-Hypnotic and Anxiolytic Drugs | Basicmedical Key
The endozepine mystery | Beyond the Ion Channel
Know Your GABA-A Receptor Subunits - by Scott Alexander
